Sri L. Menaldi
Department Of Dermatology And Venereology Faculty Of Medicine, Universitas Indonesia, Dr. Cipto Mangunkusumo General Hospital

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Journal : Jurnal MedScientiae

Inhibitor Transient Receptor Potential Vanilloid Type 1: Penggunaan Topikal pada Berbagai Dermatosis Muhammad, Parikesit; Paramitha Wibawa, Larisa; Keumala Budianti, Windy; Legiawati, Lili; Menaldi, Sri Linuwih; Rosdiana, Dewi Selvina
Jurnal MedScientiae Vol. 3 No. 2 (2024): Agustus
Publisher : Universitas Kristen Krida Wacana

Show Abstract | Download Original | Original Source | Check in Google Scholar | DOI: 10.36452/JMedScientiae.v3i2.3179

Abstract

Transient receptor potential vanilloid type 1 (TRPV1) plays an important role in the pathophysiology of pruritus and pain. TRPV1 inhibitors can reduce the sensation of itching and pain by blocking nociceptive signals from peripheral nerve fibers to the central nervous system. Topical TRPV1 inhibitors is also thought to improve skin barrier function. Therefore, TRPV1 inhibitors are considered as potential therapy in various dermatoses. Topical TRPV1 inhibitors that are currently being studied are asivatrep for atopic dermatitis and trans-4-tert-butylcyclohexanol for various dermatoses associated with sensitive skin. Further studies with better quality and longer duration are needed to assess the efficacy and safety profile of TRPV1 inhibitors.
Co-Authors Agnes Sri Siswati Ahmad Fuady Aldri Frinaldi Alida Widiawaty Anum, Qaira Aria Kekalih Augustine D. Sukarlan Bagus Haryo Kusumaputra Bani, Anna Puspitasari Caroline Oktarina Chairista, Inadia Putri Cita Rosita Sigit Prakoeswa Dewi Matindas Dewi Sumaryani Soemarko Dharmayati B. Utoyo Dhelya Widasmara Diahtantri, Riyanti Astrid Diahtantri, Riyantia Astrid Eliza Miranda Emmy Soedarmi Sjamsoe Emmy Soedarmi Sjamsoe-Daili Erika Zoulba Evita H. Effendi Fifa Argentina Fifinela Raissa Fitri Octaviana Githa Rahmayunita Hansen Angkasa Herqutanto - Hirzi Zulkarnain Irawan, Yudo Irawati, Yunia Iwan Dwiprahasto Jayawarsa, A.A. Ketut Joanne Natasha Keumala Budianti, Windy Kurniawardhani, Dewinta Retno Kusmarinah Bramono Larisa Paramitha Lidwina Anissa Lili Legiawati Lim, Henry W Lim, Henry W. Lubis, Ramona Sari Luh Karunia Wahyuni, Luh Karunia Luh Made Mas Rusyati M. Yulianto Listiawan Mamuaja, Enricco Hendra Marissa, Melani Martinus, Martinus Medhi Denisa Alinda, Medhi Denisa Melani Marissa Melani Marissa Muchtar, Vitayani Mughni, Fadhli Aulia Muhammad, Parikesit Mulianto, Nur Rachmat Olivia, Taruli Ova Emilia Rahadi Rihatmadja Regitta Indira Agusni Renni Yuniati Rizka Farah Hilma Rizky, Luddwi Achmad Rosdiana, Dewi Selvina Saleha Sungkar Sali Rahadi Asih Sandra Widaty SD, Emmy Soedarmi Sirait, Sondang Pandjaitan Siskawati, Yulia Siskawati, Yulia Sjamsoe, Emmy Soedarmi Sjamsoe-Daili, Emmy Soedarmi Surya, Denny Taruli Olivia Triana Agustin Victor Santawi Widiawaty, Alida Wresti Indriatmi B. Makes Yayi S. Prabandari Yeni Dwi Lestari Yudo Irawan Zoulba, Erika