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Journal : Journal of Pharmaceutical and Sciences.

Efektivitas Kombinasi Agen Pendeplesi Glutathione (GSH) dan Inhibitor Glutathione S-Transferase (GST) pada Resistensi Cisplatin terhadap Sel Kanker: Systematic Literature Review Nursoleha, Eva; Utami, Wahyu
Journal of Pharmaceutical and Sciences JPS Volume 8 Nomor 2 (2025)
Publisher : Fakultas Farmasi Universitas Tjut Nyak Dhien

Show Abstract | Download Original | Original Source | Check in Google Scholar | DOI: 10.36490/journal-jps.com.v8i2.777

Abstract

Cisplatin is a platinum-based chemotherapy agent used for the treatment of various types of cancer. However, the use of cisplatin as a chemotherapy agent is limited by drug resistance and side effects due to the formation of inactive metabolites from the conjugation reaction between cisplatin and Glutathione S-Transferase (GST). Thus, Glutathione (GSH) and Glutathione S-Transferase (GST) are essential in controlling cisplatin resistance. This study aims to evaluate the use of a combination of cisplatin with GSH-depleting agents and GST inhibitors to overcome or reduce cisplatin resistance in various cancer cell types in vitro and enhance cisplatin's cytotoxic activity. This research was conducted using a systematic literature review method, with a literature search across two international databases, PubMed and Science Direct, for publications from 2013 to 2024. From 15 selected journals, various GSH-depleting agents and GST inhibitors were found to improve the cytotoxic effects of cisplatin, as analyzed based on data on the levels of GSH and GST in the cells and the percentage of viable cells (% cell viability), which showed a significant decrease. The findings of this study are expected to provide insights into the development of cancer therapies using cisplatin as a chemotherapy agent.
Co-Authors Abdillah, Safira Mafaza Abdul Rahem, Abdul Abdurrahman, Zakaria Husein Adhianto, Naura Calista Adhianto Adianti, Istiana Ahsan, Dwi Adrean Aisy, Inandrohatul Ambar Yunita Nugraheni Ana Yuda Andi Suhendi Andika, Kadek Rama Andity, Vira Sekar Ayu Andry Herawati Andwini Prasetya, Andwini Andy Dwi Bayu Bawono Anindya, Talitha Ahnaf Anjaly, Ana Anjati, Yasinta Widia Antinka, Vineza Elsafa Anwar , Monica Anwar, Monica Arie Sulistyarini Arif, Hilda Meisya Arifah Sri Wahyuni Asti Arum Sari Astuti, Welly auzi, Ulfa Datrya F Azizah, Wulan Aulia Azura, Syahirah Baktiar, Bayu Balqis, Moetia Rahman Budiatin, Aniek Setiya Cholisoh, Zakky Cristian, Benny Dedi Hanwar Denny Vitasari Edelwais, Monica Eko Sumartono, Eko Erindyah Retno Wikantyasning Eriska, Ratih Erlinawati, Mira Fadhilah, Faisa Nur Fadilla, Rohayu Fauzi Ahmad Muda Fetty Chandra Wulandari Fikri, Naufal Aziz Al Firdaus, Farhand Ahmad Geri, Geri Harindasari, Amorita Azzah Heppy Purbasari Hermansyah, Andi Herri Fariadi, Herri Husna, Rozaanah Al I NYOMAN WIJAYA Ika Ratnaningrum Ika Trisharyanti Dian Kusumowati Ikrom, Muhammad Isnaniyah, Dhevi Zahra Latifatul Kaliky, Aprillia Kartikasari, Lamtana Eka Khandy, Evanda Ratna Thalia Kunnu, Hasbi Lake, Reginaldo Christopori Larasati, Arindra Liling Listyawati Lilla Puji Lestari Liza Pristianty Maharani, Laksita Umi Marijati Sangen, Marijati Mawarti, Endang Mentari Marwa, Mentari Merlindasari, Aulia Pungky Movitha, Fika Munawaroh, M Mutaqi, Ahmad Saifudin Muthiatulloh, Maryam Dzakiyah Mutmainnah, Luluk Nahrowi, Wawi Nanda S, Erika Nanditya Putra, Bramana Narda, Anya Cetta Ningtyas, Karisma Ayu Noorrizka V, Gusti Nurhadiyanti, Eva Agustin Nursoleha, Eva Nur’aini, Hesti Olivia , Dini Olivia, Dini Paradisa, Fauza Cahya Pertiwi, Aviarista Mufidah Pratama, Wahyu Putra Marga Aji Priyandani, Yuni Promono, Andreas Pujiarti, Titi Purnama Salura Puspitasari, Hanni Prihastuti Putri, Ega Annisa Rahayu, Titik Puji Rahmadani, Sandika Ramdani, Tasya Eka Regina, Tiara Ageng Ariesta Rima Munawaroh Rustiana Rustiana Safitri, Vira Saputri, Lena Sarwani Sarwani, Sarwani Setyo Nurwaini Shofiah, Mira Simanjuntak, Immanuel Binly Prima Siregar, Nia Mariana Suhardi Suhardi Sukorini, Anila Impian Syamsul Rizal Tanti Azizah Sujono Tasysaningtyas, Thalia Fiandra Tayo, Yanti Thalia Khandy, Evanda Ratna Toetik Aryani Tri Widodo, Susilo Ujiantya, Sabrina Dian Parasika Umi Athiyah, Umi Wardatul Jannah, Wardatul Wati, Abil Lia Wijaya , Afriyadi Wulandari, Risma Ayunda Yuliansyah Yuliansyah Yuliansyah Zendy Hd S, Zendy Hd S Zharifah, Jasmine Aprilia Nur Zulkamain, Bambang Subakti