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Journal : indonesian journal of pharmacy

n-Butanolic fraction of endofitic fungi of Buah Makasar increases apoptotic effect of doxorubicin on MCF-7 cells Meiyanto, Edy; Kumala, Shirly; Septisetyani, Endah Puji
Indonesian Journal of Pharmacy Vol 20 No 1, 2009
Publisher : Faculty of Pharmacy Universitas Gadjah Mada, Yogyakarta, Skip Utara, 55281, Indonesia

Show Abstract | Download Original | Original Source | Check in Google Scholar | Full PDF (664.738 KB) | DOI: 10.14499/indonesianjpharm0iss0pp42-47

Abstract

Makassar fruit, Brucea javanica (L.) Merr., showed chemopreventive activity. Secondary metabolites come from B. javanica fruit, brucatol and bruceantine, induced cell differentiation and apoptosis on Leukemia cell, while quassinoid and its derivates acted as antitumor promoter. Butanolic fraction of supernatan of endofitic fungi 1.2.11 isolate fermentation which isolated from B. javanica fruit showed cytotoxicity toward several cancer cells. This fraction has been predicted contain secondary metabolites from B. javanica and has been identified as Bruceosin and Canthin-6-one derivates. Butanolic fraction (FB) of supernatan from endofitic fungi 1.3.11 isolate fermentation is predicted for having similiar cytotoxycity as active as 1.2.11 isolate. This research is aimed to explore cytotoxycity potention dan doxorubicin on MCF-7 breast cancer cell.Synergism of BF-doxorubicin combination detect from cell viability inhibition and apoptosis induction on MCF-7, a breast cancer cell lines which shows resistancy toward doxorubicin. Cell viability on single treatment of FB and doxorubicin and its combination were carried out by MTT assay to determine IC50 and combination index (CI). Apoptosis induction of FB, doxorubicin and its combination were carried out by ethidium bromideacridine orange DNA staining.n- Butanolic fraction and doxorubicin showed cell viability inhibition on MCF-7 cell with IC50 48 μg/mL and 148 nM, respectively. Both of FB and doxorubicin showed apoptosis induction on IC50. Combination of FBdoxorubicin showed synergism and increased apoptosis induction on MCF-7 cell.Key words: Brucea javanica, endofitic fungi, MCF-7 cell, synergism, doxorubicin.
n-Butanolic fraction of endofitic fungi of Buah Makasar increases apoptotic effect of doxorubicin on MCF-7 cells Kumala, Shirly
Indonesian Journal of Pharmacy Vol 20 No 1, 2009
Publisher : Faculty of Pharmacy Universitas Gadjah Mada, Yogyakarta, Skip Utara, 55281, Indonesia

Show Abstract | Download Original | Original Source | Check in Google Scholar | DOI: 10.14499/indonesianjpharm0iss0pp42-47

Abstract

Makassar fruit, Brucea javanica (L.) Merr., showed chemopreventive activity. Secondary metabolites come from B. javanica fruit, brucatol and bruceantine, induced cell differentiation and apoptosis on Leukemia cell, while quassinoid and its derivates acted as antitumor promoter. Butanolic fraction of supernatan of endofitic fungi 1.2.11 isolate fermentation which isolated from B. javanica fruit showed cytotoxycity toward several cancer cells. This fraction has been predicted contain secondary metabolites from B. javanica and has been identified as Bruceosin and Canthin-6-one derivates. Butanolic fraction (FB) of supernatan from endofitic fungi 1.3.11 isolate fermentation is predicted for having similiar cytotoxycity as active as 1.2.11 isolate. This research is aimed to explore cytotoxycity potention and apoptosis induction of BF from 1.3.11 isolate and combination effect of BFdoxorubicinon MCF-7 breast cancer cell.Synergism of BF-doxorubicin combination detect from cell viability inhibition and apoptosis induction on MCF-7, a breast cancer cell lines which shows resistancy toward doxorubicin. Cell viability on single treatment of FB and doxorubicin and its combination were carried out by MTT assay to determine IC50 and combination index (CI). Apoptosis induction of FB, doxorubicin and its combination were carried out by ethidium bromideacridine orange DNA staining.n- Butanolic fraction and doxorubicin showed cell viability inhibition on MCF-7 cell with IC50 48 μg/mL dan 148 nM, respectively. Both of FB and doxorubicin showed apoptosis induction on IC50. Combination of FBdoxorubicin showed synergism and increased apoptosis induction on MCF-7cell.Key words: Brucea javanica, endofitic fungi, MCF-7 cell, synergism, doxorubicin.
Co-Authors . Desi . Suhaimi . Syamsudin . Yuliani Abdul Aziz Setiawan Adefira Elisyia Juniharti Adini, Syilvi Afrini Saraswati Agan Syahrial Agung Dewantoro Ahmad Subhan Aji, Nur AMEILIA AMEILIA Anarisa Budiati Andri Prasetiyo Andria Agusta Andrianopsyah Mas Jaya Putra Anggelina Aprilia Pangalila Anggi Isnaasar Anny Victor Purba Anwar Wahyudi Anwar Wahyudi Anwar, Yelfi Ariyani Kiranasari Ariyani Kiranasari Armansyah, Septiyana Lia Asnah Tarigan Atut Ruswita Atut Ruswita Handayani Aulena, Desi Nadya Aulia Tisna Dewi Ayuditiawati, Meita Bekti, Novi Dyah Purnama Bekti, Novi Dyah Purnama Carrista Carrista Dandung Ruskar Datubara, Martaulina Elisabet Delina Hasan Deni Rahmat Desi Nadya Aulena Devana Devana Dewi Laxmi Diah Dethriani Dian Indriani Dian Ratih L. Dian Ratih Laksmitawati Didik Tulus Didik Tulus Dimas Adrianto Dimas Adrianto Dosi Ahmad Yani Dwi Aryanti, Anindita Dwi Fitriyani, Dwi Dwi Hapsari Juniarti Dwi Windi Sapitri Dwi Windi Sapitri EDY MEIYANTO Elvina Dhiaul Iftitah Elvina Dhiaul Iftitah ENDRO BUDI SISWANTO Erlita Agustina Erlita Erlita Esti Mumpuni Esti Mumpuni Esti, Esti Fachry Abda El Rahman Farida, Yunahara Faridah Faridah Fauzi Setyo Fandheo Fauzia Noprima Okta Febbyasi Megawaty Gabriel Gabriel Gabriel, Gabriel Gandes Winarni Gumilar Adhi Nugroho Halim, Marta Hasan, Delina Herru Setiawan Hersunaryati, Yetti Heru Santosa Heru Santosa Hery Prambudi Hesty Utami Hesty Utami Hesty Utami R Huda, Badrul I Ketut Suada I. G.A. Ayu Wiratih Iha Haryani Hatta Iha Haryani Hatta Indah Masri Indarwati Indarwati Khairunnisa Tamimi Kurota Aini Laili Savitri Noor Lea P. Retnoningsih Leonardus B.S. Kardono Lestari Rahayu Lies Putriana Lilik Sulastri Mardiastuti, . Mardiastuti, . Marlin M. Raunsai Meiyanto, Edy Meva Sari Chandra Miftahurrohmah, Nur Mochtar, Dede Mochtar, Dede Mulatsari, Esti Muthi Ikawati Nancy Dewi Yuliana Nancy Dewi Yuliana Nancy Raisa Nancy Raisa, Nancy Noor, Laili Savitri Noviyantih, Noviyantih Nur Aji NUR ANNISA FITRI Nurmaini Nurmaini Partomuan Simanjuntak Partomuan Simanjuntak Partomuan Simanjuntak Partomuan Simanjuntak Partomuan Simanjuntak Partomuan Simanjuntak Partomuan Simanjuntak Partomuan Simanjuntak Pasanema, Dimas A. M. Pasanema, Dimas A. M. Pasaribu, Rita Kristina Peny Budiarti Pieter Hazmen Pratama, Anton Pratiwi Pujilestari Sudarmono Prih Sarnianto Prih Sarnianto Priyo Wahyudi Qodriah, Rahmatul R, Hesty Utami Rachmani, Rum Rachmani, Rum RAHMAT, DENI Raihan, Dany Ramadaniati, Hesty Utami Raymond R. Tjandrawinata Reise Manninda Restu Restiani Reubun, Yonathan Tri Atmodjo Reza Agung Sriwijaya RIRIS ISTIGHFARI JENIE Risma Marisi Tambunan, Risma Marisi Rita Kristina Pasaribu Robert Utji Rochimah Ros Sumarny RR. Ella Evrita Hestiandari Ruskar, Dandung S.Farm., M.Farm., Apt, Sondang Khairani Sarah Zaidan Sarnianto, Prih Saru Noliqo Rangkuti Sembiring, Rinawati Septisetyani, Endah Puji Sesilia A. Keban Sesilia Andriani Keban Sesilia Andriani Keban Setiadi, Feri Setiawan, Abdul Aziz Setiyarini, Setiyarini Shanny, Fransisca Shanny, Fransisca Simanjuntak, Partomuan Siswa Setyahadi Siswa Setyahadi Siswa Setyahadi Siswa Setyahadi Siswa Setyahadi Siti Jabal Mastura Sofyan Ramani Sri Widyastuti Stiani, Sofi Nurmay Sugiastuti, Fenty Suhaimi Suhaimi Suhaimi, . Syamsudin Syamsudin Syarifah Aini Syarmalina Syarmalina Teti Indrawati Teti Indrawati Umilawati Rawi Utami R, Hesty Violeta, Violeta Vyacheslav Dushenkov Wahyudi Uun Wibowo Mangunwardoyo Wida Feriningsih Widiyastuti, Asih Yati Sumiyati, Yati Yetti Hersunaryati Yonathan Atmodjo Reubun Yun Astuti Nugroho Yuniarto, Ari Yusransyah, Yusransyah