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Journal : INDONESIAN JOURNAL OF PHARMACY

THE DISSOLUTION AND DIFFUSION OF FUROSEMIDE ON SELF-NANOEMULSIFYING DRUG DELIVERY SYSTEM (SNEDDS) iis - wahyuningsih; Sugiyanto Sugiyanto; Ag. Yuswanto; Ronny Martien
Indonesian Journal of Pharmacy Vol 28 No 2, 2017
Publisher : Faculty of Pharmacy Universitas Gadjah Mada, Yogyakarta, Skip Utara, 55281, Indonesia

Show Abstract | Download Original | Original Source | Check in Google Scholar | Full PDF (699.486 KB) | DOI: 10.14499/indonesianjpharm28iss2pp112

Abstract

Furosemide a diuretic exhibits low solubility in water and low bioavailability. The purpose of this study was to determine the effect SNEDDS formation to dissolution and diffusion of furosemide. SNEDDS was made with a mixture of 66% tween 80, 26% propylene glycol, 8% oleic acid and furosemide 40mg/mL. Test for SNEDDS dissolution of the capsules was developed using USP dissolution apparatus I and compared to market products, furosemide suspenssion and furosemide powder. The medium consists of 900mL of Artificial Gastric Fluid (AGF) , phosphate buffer pH 5.8 at 37±0.5°C and stirred with a speed of 100rpm. Diffusion test of SNEDDS furosemide was conducted by using reversed rat intestinal bowel and compared to furosemide suspension and furosemide solution. The SNEDDS formulation  could enhance the dissolution and diffusion of furosemide compared to the non-SNEDDS formulation
Co-Authors Aang Gunawan Abdul Gofir Abdullah Ade Suryo Adinda Adinda Ag Yuswanto Ag. Yuswanto Agnes Dwi Wulan Mahardika Agnes Intan P.W Agung Mike Wijaya Agus Kristiyanto Agustin Tri Hastuti Agustina P. F. Seran Agustina Shinta Ahmad Ahmad Akhmad Rizal Arifudin Alexander Candra Ali Maddinsyah Ambyah Atas Aji Aminudin Aminudin Anak Agung Aris Diartama Andi Jatmiko Ani Riani Hasana Anisa Matinu Saifullah Anisatul Khoir Aprilia Anisyah Fadhillah Annas Marzuki Sulaiman Anzy Indrashanty Ardina Nilam Prawastyorini Arga Safitri Aris Santjaka Ary Kurniati Ary Kurniawati Asim Asim Ayu Trisna Dewi Az Zahro Miftakhuljanah Bambang Soepeno Bambang Supriyanto BAYU KURNIAWAN Belgiawan, Prawira Fajarindra Budi Setiyana Budy Wiryawan Cecep Pahrudin Chatarina Muryani Dadang Agus Suryanto Dedy Cahyadi Dedy Sushandoyo Denny Saputra Desyandri Desyandri dewi, fretika utami DIAN LESTARI Dikpride Despa Dina Dwi Aprilia Disman Disman Diyah Pratiwi djoko subandriyo Doddy Irawansyah Donny Kristanto Mulyantoro Dzakiyya Alya Maharani Eko Muhammad Arif Budiono Elviana R. Simbolon Emi Murniati Endra Yuliawan Endriatmo Soetarto erna wati Erti Hamimi Esensia Azama Bioasa Evy Indriasari Fadila Fitria Wulandari Fahmi Ardiansyah Faisal Amri Fajar Harianto FATIMAH FATIMAH Fatimah Fatimah Fazal Hamdan Fetty Dwi Rahmayanti Fianti Fianti Finsa Zainal Fitri Fatonah Fitria Adhi Geha Nusa Frizal Didin Mardyansyah Andita Gatot Murti Wibowo Godham Eko Saputro Gultom, Henry Casandra Guruh Prasetyo Handoko Hanik Liskustyawati, Hanik Harimukti Wandebori Harits Al Ayyubih Hasriwan Putra Hendri Hermawan Adinugraha Hendri Noviyanto Heni Ruspitasari Herawati Herawati Heri Prabowo Herma Juniati Hermanto Siregar huldan Aulia afandi Husman Husman Ibrahim, Fauzi Ida Ayu Preharsini Kusuma Iftitah Dian Humairoh Ignatius Bayu Atmoko Iis Wahyuningsih Iis Wahyuningsih Ika Putera Waspada Ilham Maulana Prihutama Ilham Wahyu Siadi Indra Iman Sumantri Inggris Yossi Pranatika Irawati Andriani Isnanik Juni Fitriyah iti Amri Alimatul Muflikhah Iwan Nurhadi Jefri Rieski Triyanto Joy Rizki Pangestu Djuansjah Kadim Kadim Kanti Rahayu Karningsih Karningsih Kayan Swastika Kayan Swatika Kirara Lena Siswanti Kusfriyadi, Mars Khendra Leny Latifah Lia Meilianingsih Liane Okdinawati Lintar Brillian Pintakami lis Wahyuningsih Lisa Andrianti Listantari Listantari Luh Putu Ratna Sundari Luthfi Ramdhansyah Lutviyah Dwi Nurfadhilah M. Choiroel Anwar Made Wena Maria Magdalena Marjono Marjono Marlia Herwening Megawati Parmasari Moh Khamim Moh Sutoro Moh. Abdul Kholik MOH. TAUFIK Moh.Taufik Mohammad Syafrizal Affandi Muchsin Doewes Mudasir Mudasir MUHAMAD RIZKI Muhammad Ba’tradiansar Muhammad Fajar Marsuki Muhammad Hanif Muhammad Reza Firmansyah Muhammad Tohir Mujiyanto Mujiyanto Nailul Himam Nana Krisdianti Nanang Sugiarto Novaria Fajar Prasetya Novie Dewi Kustiani Nugraha Nugraha Nur rohman Nuri Suryani NURULIA HIDAYAH Oktofa yudha Sudrajad Olfebri Ony Widiarto Pamungkas Pamungkas Parno Pipit Wijayanti Pranoto Pranoto Prasadja Ricardianto Pratiwi, Hasih Primadi Candra Susanto Priyono Priyono Putra, Bela Rachmat Kartolo Reslyana Dwitasari Ridho Rosmansyah Rinci Kembang Hapsari Rismi Fatoni Risna Endah Budiati Riswandi Riswandi Riszal, Akhmad Rita Noviani Rita Pasaribu Ronny Martein Ronny Martien RR. Ella Evrita Hestiandari Rubyah Hutomo Ruknan Ruknan Rully Putri Nirmala Puji Saiful Bahriyanto Sajidan Sajidan Salsabila, Unik Hanifah Santoso, Chiara Nathalie SANUSI SANUSI Sapta Kunta Purnama Sarwono Sarwono Septina Putri Bintari Singgih Prihadi Singgih Prihadi Singgih Subiyantoro Siswandari Siswandari Sitarina Widyarini Siti Amri Alimatul Muflikhah Siti Wahyuni Soesi Idayanti Sri Handayani Sri Purnami Subiakto Soekarno Suci Susanti Sudarti . Sudiyono Sudiyono Sulhadi Sulhadi Sumardi Sumardi Sumarjono Sumarjono Sumarno Sumarno Supriyono Supriyono Suryono Suryono Susy Suswaty Suwidjiyo Pramono Syafrizal Syafrizal Tarkono Tarkono Trapsilo Prihandono Tri Asih Budiati Tri Murti Andayani Tri Sakti Tunggal Dewi Tya Nur Febriana Ugeng Budi Haryoko Ujang Efendi Umiyatun hayati Triastuti Wahyu Widiyaningsih Win Akustia Win Priantoro Wira Citerawati SY, Yetti Yayan Sudaryana Yenny Puspitasari Yessi Affriyenni Yessi Gusleni Yulianti, Erni Yuswanto Yuswanto yuveline aurora zulhelmi zulhelmi