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Journal : Jurnal MIPA

Perbandingan Profil Penetrasi Formula Krim Antioksidan dari Ekstrak Perikarpium Buah Manggis (Garcinia mangostana) dengan Variasi Penetration Enhancer Siampa, Jainer Pasca; Lebang, Julianri Sari; Antasionasti, Irma; Nurmiati, Nurmiati
Jurnal MIPA Vol 10, No 1 (2021)
Publisher : Sam Ratulangi University

Show Abstract | Download Original | Original Source | Check in Google Scholar | DOI: 10.35799/jmuo.10.1.2021.31146

Abstract

Paparan sinar matahari dengan kandungan radiasi UV merupakan salah satu faktor pencetus radikal bebas penyebab penuaan dini (Photoaging), yang ditandai dengan hiperpigmentasi, kerutan, dan menurunnya elastisitas kulit. Solusi permasalahan ini adalah penggunaan antioksidan yang dapat menangkal terbentuknya radikal bebas. Tujuan dari penelitian ini adalah untuk membuat formula krim antioksidan dari ekstrak perikarpium kulit manggis dengan perbedaan penetration enhancer untuk mendapatkan persentase penetrasi dan retensi terbaik di kulit. Ekstrak perikarpium buah manggis dibuat dengan metode maserasi menggunakan etanol 70% kemudian diukur aktivitas antioksidannya dan kandungan fenoliknya, selanjutnya digunakan sebagai bahan aktif dalam formula krim. Formula F1-F3 dibuat kemudian dievaluasi karakteristik fisiknya dan dilakukan pengujian penetrasi secara in vitro. Pengujian penetrasi secara in vitro dilakukan terhadap F2 dan F3 yang mengandung ekstrak. Hasil IC50 ekstrak terhadap DPPH sebesar 7,514 µg/mL dan kandungan fenolik sebesar 112,70 ± 0,80 mgGAE/g. Nilai persentase penetrasi, persentase retensi, dan nilai flux secara berturut-turut untuk F2 sebesar 9,96% ± 0,075%; 37,951% ± 0,103%; 3,037 ± 0,023 µg/cm2.jam dan F3 sebesar 7,872% ± 0,078% ;  33,874% ± 0,259%; 2,400 ± 0,024 µg/cm2.jam. Dari hasil analisis statistik, disimpulkan bahwa F2 adalah formula terbaik dengan karakteristik fisik yang homogen, memiliki warna kekuningan, tipe emulsi m/a, pH sediaan 6, daya lekat 11,05 ± 0,87 detik, dan diameter daya sebar 6,20 ± 0,10 cm.Sun exposure with UV radiation is one of the triggers for free radicals that cause premature aging (photoaging), characterized by hyperpigmentation, wrinkles, and decreased skin elasticity. The solution to this problem is the use of antioxidants that can prevent the formation of free radicals. The purpose of this study was to formulate an antioxidant cream dosage form from pericarpium extract of mangosteen pericarpium with different penetration enhancers to obtain the best percentage of penetration and retention in the skin. Pericarpium extract of mangosteen fruit was prepared by maceration method using 70% ethanol, then the antioxidant activity and the phenolic content were measured and were used as an active ingredient in the cream formula. Formula F1-F3 were made, their physical characteristics were evaluated, and in vitro penetration testing was carried out. In vitro penetration testing was carried out on F2 and F3 containing extracts. The IC50 value of the extract against DPPH was found to be 7.514 µg/mL and the phenolic content was found to be 112,70 ± 0,80 mgGAE/g. The percentage of penetration, retention percentage, and flux value were 9.96% ± 0.075%, 37.951% ± 0.103%, 3.037 ± 0.023 µg/cm2.hour respectively for F2 and 7.872% ± 0.078% , 33.874% ± 0.259%,  2.400 ± 0.024 µg/cm2.hour, respectively for F3. From the results of statistical analysis, it was concluded that F2 was the best formula with homogeneous physical characteristics, had a yellowish color, emulsion type w/o, pH value of 6, adhesion of 11.05 ± 0.87 seconds, and diameter of spreadability of 6.20 ± 0.10 cm.
Co-Authors Abd. Kadir Abdul Hamid Abubakar, Achmad Adiaksa, Baso Witman Agus Arman, Agus Agustian Agustian Ahmad Afiif, Ahmad Ahmad Fadli AHMAD JUNAEDI Akbar Akbar Ali, St. Aminah Aminuddin Prahatama Putra Amir Amir Andriani, Reni Anik Aspirin Anissa, Fausiyah Antasionasti, Irma Anthoni Agustien Aprianti, Ulfa Apriyelita, Annisa Arie Anggraini Arnianti Arnianti Asikin, Siti Badria` Asmayani, Asmayani Asmayani, Kaswari Asmin, Risna Yunita Asriana Asriana, Asriana Audina, Zikkra Awaliah, Ainun ayu Kalista Bachtiar, Irmah Halimah Baharuddin Baharuddin Bambang Kusbandrijo Cayati, Cayati Chandra Pribadi Dahelmi Dahelmi Deswati Deswati Devin, Devin Didi Susanto, Didi Dila Fitria Dirham, Izza Fadhlinah Djunaedi Djunaedi Djurumudi J, Khairunnisa Noervaqriani Dwiani, Afe Dwisa Putra, Wahyu Efrizal Efrizal eka rahmawati Ekaningtiyas, Maya Erliza Hambali Ernawati Ernawati Fachry Abda El Rahman Faig Aizy, Fayadh Farahdiba, Syarifah Farild, Miftha Fariz Pari, Rizfi Fauzia Bakhtiar Fauziah, Ayu Bella Febrianti, Magfirah Febrianti, Mifta Fery, Fery Fettriwanti, Fettriwanti Fevria, Resti Fina Diana Firman Firman Firmansyah Firmansyah FITRAH AMALIA Fitri Deswita Fitri, Nurul Fitri, Nurwijaya G, Hasriani Gafur, Gafur Gayatri, Wulan Gazali, Zulkarnain Gustina Indriati Hadijah Hadijah Hakim, Akhmad Nur Halizah Halizah Hamansah Hamansah, Hamansah Handayani, Eka Sri Handayani, Rani Harfa, Nuraliyah Azizah Harianto, Samiin Hadi Hartati, Winda Hasan, Phika Ainnadya Hayati, Sri Ayatina Hendra, Gabriel Septian Hendrianto Hendrianto, Hendrianto Hente, Asri Hermansah Hermansah, Hermansah Hery Fajeriadi Hojang, Basri M Husnul Madihah, Husnul Hutajulu, Petrus Oktavianus Ibrahim, Muhammad Akmal Ika Aryani Ilham Ilham Intan Pramita, Intan IRA NURIYA SANTI Irawati Irawati Irma Yanti Irmawati Irmawati Irmayani Irmayani Irwan Rahman, Irwan IRWANDA, IRWANDA Isdaryanti, Isdaryanti Ismail Ismail Ismail, Wahyuni Iwan Setiawan Jadespi, Sherly Jafar, Akhmad Jannah, Siti Wardatul Jirana, Jirana Julianri Sari Lebang, Julianri Sari Jumriani, Jumriani Jusniaty, Jusniaty Kamaruddin, Muh. Ihsan Kamran, Muhammad Karim, Mutemainna Khairunnisa Khairunnisa Kiki Amelia, Kiki Kunaifi Kunaifi L, IDRUS Leli, Leli Lia Masefa, Lia Listari, Nening Lubis, Bastian Mades Fifendy Mahmudah, Yulia Nasibatul Marhaeni, Marhaeni Marwah, Syarrafah Maryana Maryana, Maryana Masrah Masrah Maya Ekaningtias Mayasari, Rini MENAUNG, FANDY Mesra Damayanti Metatia Monica Mildaratu, Mildaratu Mildawati Mildawati Mudinillah, Adam Muh. Alfi Syahrin Muhammad Arsyad Muhammad Danial Muhammad Rizaldi Trias Jaya Putra Nurdin Muhammad Sofyan Muhammad Zaini Munir, Abd. Murbayani Murbayani, Murbayani Murniati Murniati Nadiya, Zulfa Nasir, Yusrianto Nelson Nelson Nenny Indrawati, Nenny Nilah Ratnasari, Nilah Nirwana, Nirwana Nitasyawal, Mulyani Novieta, I. D. Nur Asiah Siregar Nur Faida, Nur Nurhidayah Nurhidayah Nurmina Nurmina, Nurmina Nursaeni Nursaeni, Nursaeni Nurwahyuni P, Fitriana Jufri Parhani, Aan Pariyati, Pariyati Patimang, Andi Periadnadi Periadnadi Petir Papilo Pitriyani Pitriyani Pratiwi, Aliah Puspitaloka Mahadewi, Erlina Putra, Wahyu Dwisa Putri, Adela Putri, Andi Mega Januarti Putri, Santi Diana Qudratullah, Fyzria Rahmaddiansyah, Refa Rahmah, Andi Rahman, Sari Rahayu Rahman, Suburi Rahman, Sufirman Rahmawati, Agustini Liviana Dwi Rasbawati, Rasbawati raudatul jannah Rico, Rico Ridwan, Ridwan Rijal, Abdul Rahman Khaerul Riswanti, Riswanti Risya Saputri, Risya Rita Eka Izzaty, Rita Eka Roni Jarlis Rosdeviana, Rosdeviana Rostini Rusnam Rusnam Rusti, Sukarsi Rusydi, Bahrul Ulum Sabriana, Riska Sahli, Muh Sainah, Sainah Iin Samudin, Mohammad Tofan Sanjaya sanjaya Sari, Diah Kharisma Sari, Wulan Komala Sembiring, Rinawati Septiani, Indri Sholehah, Dina Via Siampa, Jainer Pasca Siti Mariam Sjahruddin, Amran Solfiyeni Solfiyeni Srifitayani, Nur Rahma Suhartini, Eka Suhendra Suhendra Sulaeman Miru Sulistiani Sulistiani, Sulistiani Suloi, Andi Fitra Sumaryanti Sumaryanti Suparianto, Rishi Supiati Supiati Susanti Susanti Suwirmen, Suwirmen Syafrina, Vellin Putri Syamsiara Nur Syamsuddin, Naidin Taufiqqurrahman, Taufiqqurrahman Titami, Hania Tohari, Sabit TONDATUAN, ALYCIA GRACE Treasa, Adisty Dwi tri wahyuni Tri Yulianti, Tri Ula, Zumrotul Ulfiani Rahman Waddi Fatimah Wahyudi Wahyudi Wahyuningsih Wahyuningsih Wayan Kantun Widya Anggrayesti Wilna Sari Wulandari, Andi Sri Rezky Yana Ameliana Yaqutunnafis, Lale Yaumi, Ema Nuzulul Yuliati, Ni Made Yunita Kristina Yunus, Ahyuni Zakaria, Indra Junadi Zelvia Misdar Zuhri Syam Zulkarnain, A.