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LITERATURE REVIEW : Uji Molekular Docking Senyawa Osimertinib Beserta Turunannya Terhadap Reseptor Tirosin kinase Pada kanker Paru- Paru Yuliana, Dewi; Aminah, Aminah; Ishak, Andi Khuswatun Khazanah
Makassar Pharmaceutical Science Journal (MPSJ) Vol 2 No 1 (2024)
Publisher : PHARMACY UMI JOURNAL SYSTEM

Show Abstract | Download Original | Original Source | Check in Google Scholar | DOI: 10.33096/mpsj.v2i1.134

Abstract

Lung cancer is all malignancy in the lung, including malignancy originating from the lung itself (primary). In clinical terms, what is meant by primary lung cancer is a malignant tumor originating from the bronchial epithelium. Current anti-lung cancer therapy has the goal of inhibiting the activity of EGFR. One of the substances that inhibits the action of EGFR is Tyrosine Kinase Inhibitor (TKI). Osimertinib has the potential to inhibit the phosphorylation of cells containing EGFR mutations. This review article aims to determine the ability of osimertinib compounds and their derivatives as lung cancer therapeutic agents against tyrosine kinase receptors using the molecular docking method. The research method used is literature review using two databases, namely Pubmed and Google Scholar for the last 10 years from 2013-2023. And the results obtained are that Osimertinib can be used as a lung cancer therapeutic agent against tyrosine kinase receptors
Analysis of Hydroquinone in Face Whitening Cream Circulating in Pinrang Regency Mustafa, Diyan Nurkhalisah; Aminah, Aminah; Widiastuti, Harti
Makassar Pharmaceutical Science Journal (MPSJ) Vol 2 No 1 (2024)
Publisher : PHARMACY UMI JOURNAL SYSTEM

Show Abstract | Download Original | Original Source | Check in Google Scholar | DOI: 10.33096/mpsj.v2i1.172

Abstract

DIYAN NURKHALISAH M. Analysis of Hydroquinone in Face Whitening Cream Circulating in Pinrang Regency. (Supervised by Harti Widiastuti and Aminah). Whitening cream is a cosmetic preparation consisting of a mixture of chemicals and other ingredients that aims to whiten or fade black spots on the skin. Many people use whitening creams because they are sold freely. However, not all whitening creams that are sold freely are safe to use because they contain dangerous ingredients, such as hydroquinone. The purpose of this study was to analyze the hydroquinone compound in whitening cream circulating in Pinrang Regency and to find out how much hydroquinone it contained. Qualitative analysis of the four samples using the Thin Layer Chromatography (TLC) method positively contained hydroquinone which was indicated by the Rf values ​​of the samples and standard standards being the same and the appearance of purple spots which were detected under UV light of 254 nm. Quantitative analysis on four samples using the High Performance Liquid Chromatography (HPLC) method with a flow rate of 1 ml/minute, the mobile phase was methanol:aquabidestilata (55:45), the stationary phase was column C-18, the retention times of the sample and standard were obtained at the same value. namely 1.5 and 1.6 indicating that the sample contains hydroquinone. The linear regression equation y = 39.549x – 283.31 with a correlation coefficient of 0.998. The hydroquinone levels obtained were code A whitening cream of 2.5%; whitening cream B 2.8%; whitening cream C 2.45%; and whitening cream D by 0.9%.
UJI AKTIVITAS ANTIOKSIDAN EKSTRAK ETANOL KULIT PISANG RAJA (Musa paradisiaca L.) SEBAGAI BAHAN BAKU PEMBUATAN ICE CREAM DENGAN METODE FERRIC REDUCING ANTIOXIDANT POWER Abidin, Zainal; Aminah, Aminah; Ummum, Andi
Makassar Pharmaceutical Science Journal (MPSJ) Vol 1 No 4 (2024)
Publisher : PHARMACY UMI JOURNAL SYSTEM

Show Abstract | Download Original | Original Source | Check in Google Scholar | DOI: 10.33096/mpsj.v1i4.224

Abstract

Antioxidants are defined as inhibitors that work to inhibit oxidation by reacting with reactive free radicals to form stable unreactive free radicals. Antioxidants are substances that can delay, slow down and prevent the oxidation process or neutralize free radicals. Plantain peel contains several metabolite compounds that have the potential to have antioxidant activity such as saponins, polyphenols and tannins, flavonoids and terpenoids. Banana peel extract has high antioxidant activity. The methanol extract of banana peels was higher in total flavonoids and phenolics compared to the n-hexane extract of banana peels. The aim of this research was to test the antioxidant activity of the ethanol extract of plantain peel using the FRAP (Ferrc Reduxing Antioxidant Power) method. The extraction method for plantain peel uses the maceration method with 96% ethanol solvent. The ethanol extract of plantain peel was then added with several FRAP reagents then measured using a UV-Vis spectrophotometer at a wavelength of 720 nm with quercetin as a comparison and the results of the quercetin test obtained a linearity equation y = 0.0207x + 0.0114 with a correlation coefficient value of r = 0.9904. The results showed that the ethanol extract of plantain peel had antioxidant activity of 26.5828 mgQE/g extract.
Penentuan Kadar Fenolik, Tanin, Flavonoid, dan Saponin Ekstrak Etanol Daun Kenikir (Cosmos caudatus Kunth.) Abidin, Zainal; Aminah, Aminah; Razak, Rais; Eka Putri, Andi Yuyun; M, Murti Nurhidayah; A, Aridha
Makassar Pharmaceutical Science Journal (MPSJ) Vol 2 No 2 (2024)
Publisher : PHARMACY UMI JOURNAL SYSTEM

Show Abstract | Download Original | Original Source | Check in Google Scholar | DOI: 10.33096/mpsj.v2i2.249

Abstract

The kenikir plant is a tropical plant originating from Latin America that can easily grow in various places. The use of kenikir leaves (Cosmos caudatus Kunth.) as a medicinal plant has been widely used. People usually use kenikir leaves as traditional medicine. Kenikir leaves are extracted by maceration method using 96% ethanol solvent after which a liquid extract is obtained and then evaporated using a rotavapor so that a thick extract is obtained. This study aims to analyze the levels of phenolic compounds, tannins, flavonoids, and saponins contained in kenikir leaves (Cosmos caudatus Kunth.). Determination of levels using UV-Vis spectrophotometric method. The ethanol extract of kenikir leaves (Cosmos caudatus Kunth.) contains phenolic compounds, tannins, flavonoids, and saponins with the levels of each phenolic compound, tannins, flavonoids, and saponins respectively as follows: 43.592 mgGAE/g, 40.639 mgEAT/g, 36.319, and 142.527 mgSE/g.
antioxidant activity Uji aktivitas antioksidan ekstrak daun karet kebo (Ficus elastica) dengan menggunakan metode maserasi bertingkat Yani, Indah Ahmad; Suhaenah, Asriani; Aminah, Aminah
Makassar Pharmaceutical Science Journal (MPSJ) Vol 2 No 3 (2024)
Publisher : PHARMACY UMI JOURNAL SYSTEM

Show Abstract | Download Original | Original Source | Check in Google Scholar | DOI: 10.33096/mpsj.v2i3.283

Abstract

Kebo rubber (Ficus elastica) is one type of plant in Indonesia as a medicine to lower blood pressure, reduce cholesterol, stroke and reduce joint pain. In addition, Kebo rubber (Ficus elastica) leaves are one of the ficus species that are thought to be rich in polyphenolic compounds so that they can act as antioxidants. Antioxidants are compounds that can be used to counteract free radicals. Food fiber and antioxidants are two types of components that are very beneficial in improving health and being able to prevent various diseases. This study aims to analyze the antioxidant activity of rubber kebo (Ficus elastica) leaf extract using the DPPH method. The maceration process uses 3 different types of solvent, namely n-hexane (non-polae), ethyl acetate was measured at 510 nm wavelength with quercetin as the standard comparator. The measurement result for n-hexan extract obtained IC50 of 531,90 µg/mL, ethyl acetat obtained IC50 of 188,06 µg/mL, and for ethanol extract obtained IC50 of 874,73 µg/mL.
Uji Aktivitas Ekstrak Etanol Daun Kenikir (Cosmos caudatus Kunth.) Dengan Metode DPPH Abidin, Zainal; Aminah, Aminah; Sari, Nurmala
Makassar Pharmaceutical Science Journal (MPSJ) Vol 2 No 3 (2024)
Publisher : PHARMACY UMI JOURNAL SYSTEM

Show Abstract | Download Original | Original Source | Check in Google Scholar | DOI: 10.33096/mpsj.v2i3.297

Abstract

Kenikir (Cosmos caudatus Kunth.) is a traditional vegetable that can be eaten raw or cooked as a vegetable. This plant is also used for food flavoring and traditional medicine. In addition, several nutritional and medical studies show that Kenikir is rich in bioactive compounds such as flavonoids, phenols, carbohydrates, minerals, proteins and vitamins, which can increase its nutritional value. This study aims to determine the antioxidant activity of ethanol extract of kenikir leaves (Cosmos caudatus Kunth) using the DPPH method. The results showed that the ethanol extract of kenikir leaves (C. caudatus Kunth) had high antioxidant activity. Antioxidants are substances that can delay, slow down and prevent oxidation. Antioxidants are very beneficial for health and play an important role in maintaining the quality of food products. The antioxidant activity is in the very strong category (<50 ppm), namely 25,212 ppm. The macerated extract showed the highest antioxidant activity because it contained many secondary metabolites such as flavonoids and phenolics.
UJI AKTIVITAS ANTIOKSIDAN EKSTRAK ETANOL DAUN KENIKIR (Cosmos caudatus Kunth) DENGAN METODE FERRIC REDUCING ANTIOXIDANT POWER Abidin, Zainal; Salsabila Ihsan, Nur Rifdah; Aminah, Aminah
Makassar Pharmaceutical Science Journal (MPSJ) Vol 2 No 4 (2025)
Publisher : PHARMACY UMI JOURNAL SYSTEM

Show Abstract | Download Original | Original Source | Check in Google Scholar | DOI: 10.33096/mpsj.v2i4.298

Abstract

Antioxidants are defined as inhibitors that work with the oxidation process, even at relatively small concentrations. Antioxidants are substances that can delay, slow down and prevent the oxidation process. Kenikir leaves contain flavonoid compounds, polyphenols, saponins, tannins, alkaloids and essential oils and also contain bioactive compounds such as ascorbic acid, quercetin, chlorogenic acid and polyphenolic compounds which function as antioxidants. The aim of this research was to determine the antioxidant activity test of the ethanol extract of Kenikir leaves using the FRAP (Ferric Reducing Antioxidant Power) method. The Kenikir leaf extraction method uses the maceration method with 96% ethanol solvent to obtain Kenikir leaf ethanol extract. The ethanol extract of Kenikir leaves was reacted with several FRAP reagents and then measured using a UV-Vis spectrophotometer at a maximum wavelength of 720 nm. Quercetin as a comparison with the quercetin test results obtained a linearity equation of y = 0.0117x + 0.4212 with a correlation coefficient value of r = 0.9986. The results showed that the ethanol extract of Kenikir leaves had an antioxidant activity of 12.7464 mgQE/g extract.
Co-Authors A, Aridha A.A. Ketut Agung Cahyawan W Abbas, Ziana Abd. Rahim Abdillah, Nabila Sesha Abdul Aziz Abdul Fattah Abdul Haris Abdul Saman Abdullah Abdullah Abdullah Abdullah Abid, Muhammad Aditia, M. Aditiya, Syahrin Adjie , Habib Adrian Afiuddin, Lutfan Afrizal Afrizal Afrizal Nilwan Afsitin Joan Tatra Afsya, Farhan Al-Mahmudy Agripinia, Felita Agung Hartoyo Agusriyanto, Beni Ahmad Ridha Aimim-Tham, Sukanya Akbar Muchbarak Akbar, Abd. Akbar, Abdul Alamanda, Dinda Aprilia Alfi Syahrin, Alfi Aliyudin, Muhamad Amalia, Gadis amaliah, lili Ambo Ala, Ambo Amelia Sebayang Amin, Asni Amin, Lalu Yusril amir, rahmi Amir, Reski AMIRUDDIN SYAM Amri Amri Amukti, Resa Andi Irfan, Andi Andri Irawan Andriana, Riya Andriyani, Riya Anggraeni Swastika Sari Anggraeni, Bella Ani Wardah Anindita, Ivan Rifqi Anliza, Syarah Annas Boceng Appin Purisky Redaputri Aprila Niravita, Aprila Aprilianicahyati, Aprilianicahyati Aprini, Nisma Apriyani, Sri Devi Aranggraeni, Renda Ardhyarizky, Sari Ardin, Hardiani Arfan, Vina Raudhathul Arid, Muhammad Arifin, Marina Arifin, Muhammad Ahkam Arivia, Arni Ariyati, Ismi Aru Persada, I’ib Sutera Asni Amin Asriani Suhaenah Astania, Sella Erin Auliah, Nurul Awalia, Awalia Awaludin, Taufiq Ayu Septiana, Vidya Ayu, Dya Ayu, Maulida Ayuni Ayusafitri, Devita Azharuddin Azharuddin, Azharuddin Azyurah, Zilmi B, Irwan Bachrul Amiq Badu, Nurul Fadillah Bangun Wijonarko, Bangun Basri, Lambang Bastiana Bastiana Betty Magdalena, Betty Bidhari, Lesty Ayu Bintang, Dinantara Mega Birton, Salzavira Belliananda Borman, M. Syahrul Budhi Waskito Budi Ispriyarso Budiyanti, Fitriyani Bunga, A. Tenri Busaeri, St. Rahbiah Dagong, Muh. Ihsan A. Danu Virgiawan, Fazar Desiana, Wahdah Desrin Lebagi Devega, Meta Devira Utami, Herdiyanti Dewi Lokida Dewi Sartika Munthe Dewi Yuliana Dewi, Anjar Kusuma dian mega putri, dian mega Dinata Pemuka, Riska Dindasari, Dita Djaya, Ernawati Doddy Ismunandar Bahari Dongoran, Hana Marty Eddy, Syaiful Edy Edy Effendi Hasan Efriyanto, Efriyanto Eka Fitriani Eka Putri, Andi Yuyun Eka Sri Handayani Eli Amaliyah Endang Pratiwi4, Endang Pratiwi4 Erfiani Erfiani Ernawati Ernawati Ervina, Iin Ery Agus Priyono, Ery Agus Evi Gantyowati Fadel, Muh. Fadel, Muhammad Fadillah, Minda Fadjry Djufry Farial Farial Farial, Nur Hasanah Fathurohman, I Fatmawati Fatmawati FAUSIAH, FAUSIAH Febriana, Michelle Fellisia, Mega Fifiana Wisnaeni Finte Nate, Aisya Firdaus Firdaus Firdaus, Firdianti Firmansyah, Doni Fitri, Nurul Futri, Elisa Futri Gemini, Pra Grace Nathalie, Giftania Grace Novenasari Manurung Graisman.P, Naufal Grazetta, Vicko Vanessa Hafizha, Tsaniya Haji Hamil, Haji Jamaie Hamsinah Hamsinah, Hamsinah Handayani, Fitriana Haninun Hapsari, Shabrina Haq, Sadida Amalia Izzatul Harahap, Mira Apriani Harauly Lady Lusiana Manalu Hardiyansyah Hardiyansyah Hardiyanti, Marzellina Hari Prihanto, Purwaka HARI PURNOMO Hartabela, Dadang Harti Widiastuti Hartina, Suki Hasbi Hasnaeni hasnaeni, Hasnaeni Hasyim, Moh. Yusuf Ahmad Hendra, Aldi Alma Hendri Hendri Henny Murtini Herawati Herawati Herlina Herlina Herman, Widyawati Herni Widanarti Hidayatullah, Muhammad Zamroni Hizbullah, Auliya Holida, Ida Huda, Syariful Husnaeni Husnaeni Husnul Madihah I Nyoman loka Ibrahim, Elisurya Ida Suryani, Ida Ida Syafrida Ihsan, Muhammad Taufik Ike Puspasari Ayu Ilyas, Mohd Imam Himawan Imam Machali Imanuriea Annisa Putri Indradewa, Rhian Indrati Rini, Indrati Irawati Irawati Irma Cahyaningtyas, Irma Ishak, Andi Khuswatun Khazanah Iskandar Zulkarnain, Ali Iskandar, Rina Ismaniar Ismaniar Ismayanti, Rini Jamiluddin, Jamiluddin Jarkawi Jolianis ME S.Pd Julaeha, Eha Julailah, Julailah Juliana, Putri Kaban, Fitriyana Br Kaimuddin Kaimuddin, Kaimuddin Kamaruddin , Abdul Kamaruddin, Abd Kanzunnudin, M Kapura Sary, Dwi Karlina Syahruddin, Karlina Khair, Oki Iqbal Khairudin Khairudin Khairunnisa, Indah Khalda, Hanindya Naufal Khalda, Nabila khusnul khotimah Konder Manurung Kuntoro, Brama Kurnaliah, Kurnaliah Kusmita, Riya L. Lisnawati Laelatul Anisah, Laelatul Lahmi, Ahmad Latifah, Rosiana Laudza, Kamelia Anis Listia Wati, Nur Luke Suciyati Amna Lukis Alam M Atik Martiningsih, M Atik M, Murti Nurhidayah Madaskolay Viktoris Dahoklory Maf'ulah, Maf’ulah Maghfira Faraidiany Mahagiyani, Mahagiyani Mahara, Emi Mahara, Husnah Mahsup, Mahsup Maisura Maisura Mamat Pratama, Mamat Mardiyah, Nur Margaretha, Nina Vernia Maria, Anna Marisa Marisa Masdiana Tahir Mashuri Mashuri Masnawati Masnawati, Masnawati Mauli, Izaton Mayang Sari, Silviana MAYUASTI MAYUASTI Meidina, Tatiana Melana, Lilis Meldilianus N J Lenas Meredian Alam Miranda, Yula Mochamad Hadi Mochtar Marhum Mohzana Monica Marpaung, Dorima Muammar Fawwaz Muchamad Subali Noto Muhammad Azmi, Muhammad Muhammad Fadhil Muhammad Muhammad Muhammad Reza Muhammad Rizal Fadilah Muhammad, Faik Muharni Muharni Muharram, Muhammad Fikri Mujtahid, Izzatul Fikri Mukhrijal Mukhrijal Mukrim, Mukrim Muliadi, Mus Munandar, Surahmat Agus Muntari Muntari Mustafa, Diyan Nurkhalisah Mustajab, Duta Musthofa, Imron Mutiara, Ravika Najamuddin, Erwin Nasaruddin Nasaruddin Nasution, Nurjannah Ni Putu Widhia Rahayu Ningrum, Karmila Ningsih, Resty Setia Nisa, Khaerun Noermalita, Azahra Mona Noventi, Endiyah Novidawati Boru Situmorang Novita Sari Nugraheni Nugraheni Nur Aliyah Nur, Nur Aliyah Nur Annisa, Akrima Nur Rahmi, Maulida Anggun Nur, Aprisal Nur, Fenty Nurachmawaty, Nabillah Nuraeni Nuraeni Nuranisah, Nuranisah Nurazima, Nurazima Nurdia, Nurdia Nurdiawansyah Nurhasanah, Lisa Nurliadi, Indah Nurlisa Nurlisa Nurmala Sari Nurul Fuadi Oktalivia, Ardhita Oktaviani, Marsella Orowala, Anggriani Padjung, Rusnadi Palad, Marliana S Palad, Marliana S. Pangestu, Aditya Paramita Prananingtyas Pebrianti, Novi Pernando, Anggra Pohan, Nurhikmah Prastyanto, Yusman Pratiwi, Endang Pratiwi Priyanto, Slamet Bambang PUDJI ASTUTI Purbaningsih, Yuli Putri Ratna Sari, Putri Ratna Putri, Dwi Adhinda Junaidi Putri, Hapshah Azzahra Welvi Putri, Jennie Calista Putri, Ryzkya Amanda Qadaruddin Fajri Adi Qawiy, Haqi Romadhona Rachmawati, Fairus Augustina Rachmawati, Nurmeily Rahmaini Fitri Harahap Rahman Rahman Rahman, Ayyub Ar Rahmawan, Mohammad Iqbal Rahmi Wahyuni, Rahmi Rais Razak, Rais ramadhan, nurhaliza Ramadini, Ristieyen Raodatul Jannah Ratnawati Ratnawati Rekhan. T, Muh Rafli Renny Mointi Retnoningrum, Jasmine Aryanti Revaldy, Muhammad Arsy Ridwan, Nur Fathurahman Ridwansyah , M. Rina Iskandar Rinitami Njatrijani Ririn Risda Waris, Risda Riska Riska Rizki, Sari Rizky, Fahim Muhammad Robbo, Anwar Rochman, Auliya Romaulianna Theresia Marbun Rosya, Dianda Talitha Rowina, Sinta Roy Efendi, Roy Rudi Haryadi, Rudi Rusmin Nuryadin Sabahannur, St Sabit Tohari Safira, Mutiarasafira Sahur, Asmiaty Saida, dan Saipul Abbas Salam, La Ode Muh. Aswad Salpina . Salsabela, Ghina Salsabila Ihsan, Nur Rifdah Samparan, Nirwana Sandyna, Muhammad Ivan Saniasa, Saniasa Sanjaya sanjaya Saputra, Meli Saputra, Pijai Opin Saputra, Reshar Saputri, Nur Airin Saragih, Elv. Feedia Mona Sardani, Rama Aditiya Sari, Yuli Eka Sarmawi, Sarmawi Sarwo, Yohanes Budi Sastra, Satrian Sawal, An-nafi Selpida Handayani, Selpida Seniwati Seniwati, Seniwati Septiandi, Dian Ayu Shafiyuddin, Muhammad Shelviani, Hanasa Siahaan, Gelora Chita Sigit Budi Santoso, Sigit Budi Silvi Listia Dewi Sinaga, Elvina Sari sipi, Surianto Siregar, Ryskina Fatimah Siti Fatimah Siti Hadijah SITI MARYAM Siti Nurhayati Siti Rahmawati Siti Sunariyati Soleha Soleha Sopian sopian Sri Ayatina Hayati Sri Ernawati Sri Mulyani Sri Wahyuni Sriati Usman St. Maryam, St. St. Sabahannur Suari, Ine Suci Ramadhani, Suci Sudamara, Yamon Sudirman Numba Sugianto, Fitri Alina Sugiono Sugiono Sugito - Sukma, Zhilla Permata Radela Sunarjati, Sunarjati Suwandi Suwandi Suwardi Suwardi Syafadila, Elva Syafadilla, Elva Syahdar Baba Syam, Netty Syarief, Faisal Syarif Prakoso, Ramzy Tadjuddin Naid Taliding, Arianto Taufik, Moh Tina Miniawati Barusman Tony, Frans Tri Damayanti Tri Widayatsih, Tri Trisna, Citra Tristy, Marsatana Tartila Tursina Tursina Ubaidullah Ubaidullah, Ubaidullah Ubaidulllah, Ubaidulllah Ummum, Andi Utami, Anita Syafira Utami, Riyandini Riyan Verawaty Fitrinelda Silaban Vicha Hulai, Bella Wahdini, Wahdini Wahyudi, Mochammad Rezza Wahyudin Wahyudin Wahyuni, Ayusari Wati, Wahyuni Kencana Wibowo, Rifdah Oktavia Wildan Wildan Winarna, Jaka Wulandari, Ghina Antania Yani, Indah Ahmad Yani, Sefty Yenni Del Rosa Yuliani, RA Dewi Maria Yumna, Lonita Aini YUNUS MUSA Yusliza, Yusliza Yusriana Yusriana, Yusriana Yusriani, Yusriani Yusrimuddin, Yusrimuddin Yusriyadi Yusriyadi Zaenudin Zaenudin Zahriyanti Zainal Abidin Zelviani, Sri Zukhaira - Zulfikar Husni Faruq Zuliani, Tiara Destika